By Xiao-Tian Liang, Wei-Shuo Fang
Present discoveries and learn into bioactive common products
Medicinal Chemistry of Bioactive average items presents a much-needed survey of bioactive usual items and their functions in medicinal chemistry. This accomplished reference positive aspects articles through many of the world's top scientists within the box on discovery, constitution elucidation, and stylish man made strategies--developed for usual products--with an emphasis at the constitution job courting of bioactive normal items. the themes were rigorously selected at the foundation of relevance to present study and to value as clinicially valuable agents.
instead of trying to be a accomplished encyclopedia of bioactive average items, Medicinal Chemistry of Bioactive usual items publications the reader to the main advancements within the box. by way of delivering not just useful element yet a old standpoint at the chemistry and biology of the compounds into consideration, the ebook serves as a convenient source for researchers of their personal paintings constructing prescribed drugs, and as an inspiring advent for younger scientists to the dynamic box of bioactive ordinary items research.
better by way of examples with up-to-date study effects, the dialogue covers such themes as:
* The chemistry and biology of epothilones
* Vancomycin and different glycopeptide antibiotic derivates
* Antitumor and different comparable actions of Taxol and its analogs
* The antimalarial homes of the normal chinese language drugs, Quinghaosu (artemisinin)
* Huperzine A: A usual drug for the therapy of Alzheimer's disease
* The medicinal chemistry of ginkgolides from Ginkgo biloba
* contemporary development in Calophyllum coumarins as effective anti-HIV agents
* Plant-derived anti-HIV brokers and analogs
* Chemical synthesis of annonaceous acetogenins and their structurally changed mimics
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